Discovery of a New Class of Potent MMP Inhibitors by Structure-Based Optimization of the Arylsulfonamide Scaffold-Reference-Cited by-同舟云学术

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Discovery of a New Class of Potent MMP Inhibitors by Structure-Based Optimization of the Arylsulfonamide Scaffold

Published:2013-05-14 Issue:6 Volume:4 Page:565-569
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Mori Mattia¹²,Massaro Assunta¹,Calderone Vito²,Fragai Marco²³,Luchinat Claudio²³,Mordini Alessandro⁴

Affiliation:

1. ProtEra Srl, Scientific Campus, University of Florence, viale delle idee 22, I-50019 Sesto Fiorentino, Italy

2. Magnetic Resonance Center (CERM), University of Florence, via L. Sacconi 6, I-50019 Sesto Fiorentino, Italy

3. Department of Chemistry “Ugo Shiff”, University of Florence, via della Lastruccia 3, I-50019 Sesto Fiorentino, Italy

4. ICCOM-CNR, Dipartimento di Chimica “U. Schiff”, via della Lastruccia 13, I-50019 Sesto Fiorentino, Italy

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml300446a

Reference31 articles.

1. Predicting the Binding Mode of Known NCp7 Inhibitors To Facilitate the Design of Novel Modulators

2. Simple Pseudo-dipeptides with a P2′ Glutamate

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2. Structural analysis of arylsulfonamide-based carboxylic acid derivatives: a QSAR study to identify the structural contributors toward their MMP-9 inhibition;Structural Chemistry;2020-09-17

3. Molecular modeling and biological studies show that some μ-opioid receptor agonists might elicit analgesia acting as MMP-9 inhibitors;Future Medicinal Chemistry;2019-06

4. An integrated structure- and pharmacophore-based MMP-12 virtual screening;Molecular Diversity;2018-02-08

5. Design, synthesis, SAR and biological investigation of 3-(carboxymethyl)rhodanine and aminothiazole inhibitors of Mycobacterium tuberculosis Zmp1;Bioorganic & Medicinal Chemistry Letters;2018-02

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