From Phenothiazine to 3-Phenyl-1,4-benzothiazine Derivatives as Inhibitors of the Staphylococcus aureus NorA Multidrug Efflux Pump-Reference-Cited by-同舟云学术

From Phenothiazine to 3-Phenyl-1,4-benzothiazine Derivatives as Inhibitors of the Staphylococcus aureus NorA Multidrug Efflux Pump

Published:2008-06-25 Issue:14 Volume:51 Page:4321-4330
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sabatini Stefano¹,Kaatz Glenn W.¹,Rossolini Gian Maria¹,Brandini David¹,Fravolini Arnaldo¹

Affiliation:

1. Dipartimento di Chimica e Tecnologia del Farmaco, Università di Perugia, 06123 Perugia, Italy, Department of Internal Medicine, Division of Infectious Diseases, School of Medicine, Wayne State University and the John D. Dingell Department of Veterans Affairs Medical Center, Detroit, Michigan 48201, USA, Dipartimento di Biologia Molecolare, Laboratorio di Fisiologia e Biotecnologia dei Microrganismi, Università di Siena, 53100 Siena, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm701623q

Reference70 articles.

1. New strategies for combating multidrug-resistant bacteria

2. Proton-dependent multidrug efflux systems.

3. Antiseptic susceptibility and distribution of antiseptic-resistance genes in methicillin-resistantStaphylococcus aureus

4. Bacterial enzymatic resistance: β-lactamases and aminoglycoside-modifying enzymes

5. Erythromycin resistance by ribosome modification

Cited by 104 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis, X-ray, spectroscopic characterizations, DFT calculations, Hirschfeld surface analyses, molecular docking, and molecular dynamic simulations of some 1,4-benzothiazine-1,1-dioxide derivatives as human kinase CK2 inhibitors;Journal of Molecular Structure;2024-09

2. Unraveling the ligand specificity and promiscuity of the Staphylococcus aureus NorA efflux pump: a computational study;Journal of Biomolecular Structure and Dynamics;2024-03-18

3. Potential anti-amoebic effects of synthetic 1,4-benzothiazine derivatives against Acanthamoeba castellanii;Heliyon;2024-01

4. Recent developments in the synthesis of hybrid heterocycles, a promising approach to develop multi-target antibacterial agents;Journal of Molecular Structure;2023-08

5. Fighting Antimicrobial Resistance: Insights on How the Staphylococcus aureus NorA Efflux Pump Recognizes 2-Phenylquinoline Inhibitors by Supervised Molecular Dynamics (SuMD) and Molecular Docking Simulations;Journal of Chemical Information and Modeling;2023-07-29