Synthesis of a Novel Macrocyclic Library: Discovery of an IGF-1R Inhibitor-Reference-Cited by-同舟云学术

Synthesis of a Novel Macrocyclic Library: Discovery of an IGF-1R Inhibitor

Published:2008-02-14 Issue:2 Volume:10 Page:256-266
ISSN:1520-4766
Container-title:Journal of Combinatorial Chemistry
language:en
Short-container-title:J. Comb. Chem.

Author:

Qvit Nir¹,Reuveni Hadas¹,Gazal Sharon¹,Zundelevich Adi¹,Blum Galia¹,Niv Masha Y.¹,Feldstein Alexandra¹,Meushar Sharon¹,Shalev Deborah E.¹,Friedler Assaf¹,Gilon Chaim¹

Affiliation:

1. Department of Organic Chemistry, Department of Biological Chemistry, Department of Physical Chemistry, The Fritz Haber Research Center, and The Wolfson Centre for Applied Structural Biology, The Hebrew University of Jerusalem, Jerusalem 91904, Israel

Publisher

American Chemical Society (ACS)

Subject

General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cc700113c

Reference53 articles.

1. Target-Oriented and Diversity-Oriented Organic Synthesis in Drug Discovery

2. Applications of Combinatorial Technologies to Drug Discovery. 1. Background and Peptide Combinatorial Libraries

3. Solution- and Solid-Phase Strategies for the Design, Synthesis, and Screening of Libraries Based on Natural Product Templates: A Comprehensive Survey

4. Compounds That Activate the Mouse Melanocortin-1 Receptor Identified by Screening a Small Molecule Library Based upon the β-Turn

5. β-Turn mimetic library synthesis: scaffolds and applications

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