Structure−Activity Relationship of Small-Sized HIV Protease Inhibitors Containing Allophenylnorstatine-Reference-Cited by-同舟云学术

Structure−Activity Relationship of Small-Sized HIV Protease Inhibitors Containing Allophenylnorstatine

Published:1999-04-24 Issue:10 Volume:42 Page:1789-1802
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mimoto Tsutomu¹,Kato Ryohei¹,Takaku Haruo¹,Nojima Satoshi¹,Terashima Keisuke¹,Misawa Satoru¹,Fukazawa Tominaga¹,Ueno Takamasa¹,Sato Hideharu¹,Shintani Makoto¹,Kiso Yoshiaki¹,Hayashi Hideya¹

Affiliation:

1. Pharmaceuticals & Biotechnology Laboratory, Japan Energy Corporation, Toda-shi, Saitama 335-8502, Japan, and Department of Medicinal Chemistry, Kyoto Pharmaceutical University, Yamashina-ku, Kyoto 607-8414, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm980637h

Reference28 articles.

1. Endoproteolytic cleavage of gp160 is required for the activation of human immunodeficiency virus

2. Current Status of the Development of HIV Protease Inhibitors and Their Clinical Potential

3. Kynostatin (KNI-227 and -272, highly potent anti-HIV agents: conformationally constrained tripeptide inhibitors of HIV protease containing allophenylnorstatine.

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