Structure-Based Design of 2-Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors-Reference-Cited by-同舟云学术

Structure-Based Design of 2-Aminopyridine Oxazolidinones as Potent and Selective Tankyrase Inhibitors

Published:2013-10-23 Issue:12 Volume:4 Page:1218-1223
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Huang Hongbing¹,Guzman-Perez Angel¹,Acquaviva Lisa¹,Berry Virginia¹,Bregman Howard¹,Dovey Jennifer¹,Gunaydin Hakan¹,Huang Xin¹,Huang Liyue¹,Saffran Doug¹,Serafino Randy¹,Schneider Steve¹,Wilson Cindy¹,DiMauro Erin F.¹

Affiliation:

1. Departments of Medicinal Chemistry; ‡Pharmacokinetics and Drug Metabolism; §Oncology Research; and ∥Molecular Structure, Amgen Inc., 360 Binney Street, Cambridge, Massachusetts 02142, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml4003315

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