Chemical and Biological Investigation of Cyclopropyl Containing Diaryl-pyrazole-3-carboxamides as Novel and Potent Cannabinoid Type 1 Receptor Antagonists
Author:
Affiliation:
1. Medicinal Chemistry Research Laboratory IV, Gedeon Richter Plc, PO Box 27, H-1475 Budapest 10, Hungary
2. Division of Drug Safety and Pharmacology, Gedeon Richter Plc, PO Box 27, H-1475 Budapest 10, Hungary
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm900179y
Reference38 articles.
1. Obesity: The Disease
2. The extent of the problem of obesity
3. Obesity as a risk factor for cardiovascular disease
4. Management of Obesity in Adults: European Clinical Practice Guidelines
5. Obesity: an epidemic in need of therapeutics
Cited by 34 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Copper-Promoted Aerobic Oxidative [3+2] Cycloaddition Reactions of N,N-Disubstituted Hydrazines with Alkynoates: Access to Substituted Pyrazoles;The Journal of Organic Chemistry;2023-02-01
2. Synthesis of pyrazoles from sulfonyl hydrazone and benzyl acrylate under transition-metal-free conditions;Organic & Biomolecular Chemistry;2023
3. A Regioselective Synthesis of 5-chloro-1-vinyl- and 3-alkenyl-5-chloro-1H-pyrazoles;Chemistry of Heterocyclic Compounds;2022-11
4. Synthesis of Pyrazole Compounds by Using Sonication Method;Oriental Journal Of Chemistry;2022-02-28
5. Base promoted CuFe 2 O 4 catalyzed one‐pot synthesis of 3, 5‐diaryl‐1 H ‐pyrazoles;Journal of Heterocyclic Chemistry;2021-11-10
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3