High-Resolution Crystal Structures of Human Cyclin-Dependent Kinase 2 with and without ATP: Bound Waters and Natural Ligand as Guides for Inhibitor Design-Reference-Cited by-同舟云学术

High-Resolution Crystal Structures of Human Cyclin-Dependent Kinase 2 with and without ATP: Bound Waters and Natural Ligand as Guides for Inhibitor Design

Published:1996-01-01 Issue:23 Volume:39 Page:4540-4546
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Schulze-Gahmen Ursula¹,De Bondt Hendrik L.¹,Kim Sung-Hou¹

Affiliation:

1. Department of Chemistry and Lawrence Berkeley National Laboratory, University of California, Berkeley, California 94720, and Faculteit Farmaceutische Wetenschappen, Laboratorium voor Analytische Chemie en Medicinale Fysicochemie, K. U. Leuven, E. Van Evenstraat 4, B-3000 Leuven, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960402a

Reference32 articles.

1. The Protein Kinase Family: Conserved Features and Deduced Phylogeny of the Catalytic Domains

2. Diversity in function and regulation of MAP kinase pathways

3. MAPKs: new JNK expands the group

4. Specificity of receptor tyrosine kinase signaling: Transient versus sustained extracellular signal-regulated kinase activation

5. Signal transduction and growth control in yeast

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