Aminopiperidine Sulfonamide Cav2.2 Channel Inhibitors for the Treatment of Chronic Pain-Reference-Cited by-同舟云学术

Aminopiperidine Sulfonamide Cav2.2 Channel Inhibitors for the Treatment of Chronic Pain

Published:2012-11-12 Issue:22 Volume:55 Page:9847-9855
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Shao Pengcheng P.¹,Ye Feng¹,Chakravarty Prasun K.¹,Varughese Deepu J.¹,Herrington James B.²,Dai Ge²,Bugianesi Randal M.²,Haedo Rodolfo J.²,Swensen Andrew M.²,Warren Vivien A.²,Smith McHardy M.²,Garcia Maria L.²,McManus Owen B.²,Lyons Kathryn A.³,Li Xiaohua³,Green Mitchell³,Jochnowitz Nina⁴,McGowan Erin⁴,Mistry Shruti⁴,Sun Shu-Yu⁴,Abbadie Catherine⁴,Kaczorowski Gregory J.²,Duffy Joseph L.¹

Affiliation:

1. Departments of Medicinal Chemistry, Merck Research Laboratories, Rahway, New Jersey 07065, United States

2. Ion Channels, Merck Research Laboratories, Rahway, New Jersey 07065, United States

3. Drug Metabolism and Pharmacokinetics, Merck Research Laboratories, Rahway, New Jersey 07065, United States

4. Pharmacology, Merck Research Laboratories, Rahway, New Jersey 07065, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301056k

Reference30 articles.

1. Contemporary Management of Neuropathic Pain for the Primary Care Physician

2. Intrathecal Therapy: What Has Changed With the Introduction of Ziconotide

3. Pre- and postsynaptic contributions of voltage-dependent Ca2+ channels to nociceptive transmission in rat spinal lamina I neurons

4. Structure and Functional Expression of an ω-Conotoxin-Sensitive Human N-Type Calcium Channel

5. Use-dependent blockade of Cav2.2 voltage-gated calcium channels for neuropathic pain

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