Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as Potent Carbonic Anhydrase Inhibitors: Synthesis, Biological Evaluation, and Enzyme−Ligand X-ray Studies-Reference-Cited by-同舟云学术

Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as Potent Carbonic Anhydrase Inhibitors: Synthesis, Biological Evaluation, and Enzyme−Ligand X-ray Studies

Published:2010-02-19 Issue:6 Volume:53 Page:2401-2408
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Gitto Rosaria¹,Agnello Stefano¹,Ferro Stefania¹,De Luca Laura¹,Vullo Daniela²,Brynda Jiri³⁴,Mader Pavel³⁴,Supuran Claudiu T.²,Chimirri Alba¹

Affiliation:

1. Dipartimento Farmaco-Chimico, Università di Messina, Viale Annunziata, I-98168 Messina, Italy

2. Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Firenze, Italy

3. Department of Structural Biology, Institute of Molecular Genetics, Academy of Sciences of the Czech Republic, CZ-16637 Prague, Czech Republic

4. Department of Structural Biology, Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic, CZ-16637 Prague, Czech Republic

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9014026

Reference58 articles.

1. Carbonic Anhydrase Inhibitors as Anticonvulsant Agents

2. Carbonic anhydrase inhibitors as emerging drugs for the treatment of obesity

3. Carbonic Anhydrase Inhibitors and the Management of Cancer

4. Carbonic anhydrase inhibitors

5. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

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