Synthesis and Pharmacological Evaluation of Triflate-Substituted Analogues of Clozapine: Identification of a Novel Atypical Neuroleptic-Reference-Cited by-同舟云学术

Synthesis and Pharmacological Evaluation of Triflate-Substituted Analogues of Clozapine: Identification of a Novel Atypical Neuroleptic

Published:1997-12-01 Issue:25 Volume:40 Page:4146-4153
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Liao Yi¹,DeBoer Peter¹,Meier Eddie¹,Wikström Håkan¹

Affiliation:

1. Department of Medicinal Chemistry, University of Groningen, A. Deusinglaan 1, NL-9713 AV, Groningen, The Netherlands, and Lundbeck A/S, Ottiliavej 9, DK-2500, Copenhagen-Valby, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9704457

Reference54 articles.

1. Dopamine Receptor Binding Predicts Clinical and Pharmacological Potencies of Antischizophrenic Drugs

2. Antipsychotic drug doses and neuroleptic/dopamine receptors

3. Antagonism by neuroleptics of neurotransmitter receptors of normal human brain in vitro

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