Kinase Inhibitor Data Modeling and de Novo Inhibitor Design with Fragment Approaches
Author:
Affiliation:
1. Eli Lilly and Company Lilly Research Laboratories, Lilly Corporate Center, DC 1931, Indianapolis, Indiana 46285
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm901147e
Reference33 articles.
1. Therapeutic Protein Kinase Inhibitors
2. A small molecule–kinase interaction map for clinical kinase inhibitors
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4. Characteristic Physical Properties and Structural Fragments of Marketed Oral Drugs
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