Development of an Efficient Pd-Catalyzed Coupling Process for Axitinib-Reference-Cited by-同舟云学术

Development of an Efficient Pd-Catalyzed Coupling Process for Axitinib

Published:2013-06-07 Issue:1 Volume:18 Page:266-274
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Chekal Brian P.¹²,Guinness Steven M.¹²,Lillie Brett M.¹²,McLaughlin Robert W.¹²,Palmer Charles W.¹²,Post Ronald J.¹²,Sieser Janice E.¹²,Singer Robert A.¹²,Sluggett Gregory W.¹²,Vaidyanathan Rajappa¹²,Withbroe Gregory J.¹²

Affiliation:

1. Chemical Research and Development, Pfizer Worldwide Research and Development, Groton Laboratories, Eastern Point Road, Groton, Connecticut 06340, United States

2. Analytical Research and Development, Pfizer Worldwide Research and Development, Groton Laboratories, Eastern Point Road, Groton, Connecticut 06340, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op400088k

Reference36 articles.

1. Vascular Endothelial Growth Factor as a Target for Anticancer Therapy

2. Nonclinical Antiangiogenesis and Antitumor Activities of Axitinib (AG-013736), an Oral, Potent, and Selective Inhibitor of Vascular Endothelial Growth Factor Receptor Tyrosine Kinases 1, 2, 3

3. bKania, R. S.; Bender, S. L.; Borchardt, A. J.; Braganza, J. F.; Cripps, S. J.; Hua, Y.; Johnson, M. D.; Johnson, T. O., Jr.; Luu, H. T.; Palmer, C. L.; Reich, S. H.; Tempczyk-Russell, A. M.; Teng, M.; Thomas, C.; Varney, M. D.; Wallace, M. B.PCT Int. Appl. WO/2001/002369, 2001.

4. Comparative effectiveness of axitinib versus sorafenib in advanced renal cell carcinoma (AXIS): a randomised phase 3 trial

5. The Heck Reaction as a Sharpening Stone of Palladium Catalysis

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