Bidirectional, Iterative Approach to the Structural Delineation of the Functional “Chemoprint” in GPR40 for Agonist Recognition-Reference-Cited by-同舟云学术

Bidirectional, Iterative Approach to the Structural Delineation of the Functional “Chemoprint” in GPR40 for Agonist Recognition

Published:2007-06-01 Issue:13 Volume:50 Page:2981-2989
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tikhonova Irina G.¹,Sum Chi Shing¹,Neumann Susanne¹,Thomas Craig J.¹,Raaka Bruce M.¹,Costanzi Stefano¹,Gershengorn Marvin C.¹

Affiliation:

1. Laboratory of Biological Modeling, Clinical Endocrinology Branch, Chemical Biology Core Facility, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0614782

Reference53 articles.

1. Computational Modeling Approaches to Structure−Function Analysis of G Protein-Coupled Receptors

2. Molecular mechanisms of ligand binding, signaling, and regulation within the superfamily of G-protein-coupled receptors: molecular modeling and mutagenesis approaches to receptor structure and function

3. Historical review: A brief history and personal retrospective of seven-transmembrane receptors

4. Techniques: Recent developments in computer-aided engineering of GPCR ligands using the human adenosine A3 receptor as an example

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