Selective Agonists at Group II Metabotropic Glutamate Receptors: Synthesis, Stereochemistry, and Molecular Pharmacology of (S)- and (R)-2-Amino-4-(4-hydroxy[1,2,5]thiadiazol-3-yl)butyric Acid-Reference-Cited by-同舟云学术

Selective Agonists at Group II Metabotropic Glutamate Receptors: Synthesis, Stereochemistry, and Molecular Pharmacology of (S)- and (R)-2-Amino-4-(4-hydroxy[1,2,5]thiadiazol-3-yl)butyric Acid

Published:2002-08-13 Issue:19 Volume:45 Page:4240-4245
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Clausen Rasmus P.¹,Bräuner-Osborne Hans¹,Greenwood Jeremy R.¹,Hermit Mette B.¹,Stensbøl Tine B.¹,Nielsen Birgitte¹,Krogsgaard-Larsen Povl¹

Affiliation:

1. NeuroScience PharmaBiotec Research Center, Department of Medicinal Chemistry, The Royal Danish School of Pharmacy, 2 Universitetsparken, DK-2100 Copenhagen, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020122x

Reference39 articles.

1. Ligands for Glutamate Receptors: Design and Therapeutic Prospects

2. Molecular determinants of metabotropic glutamate receptor signaling

3. Glutamate in CNS disorders as a target for drug development: an update

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