10-Substituted 11-Oxygenated (R)-Aporphines: Synthesis, Pharmacology, and Modeling of 5-HT1A Receptor Interactions-Reference-Cited by-同舟云学术

10-Substituted 11-Oxygenated (R)-Aporphines: Synthesis, Pharmacology, and Modeling of 5-HT1A Receptor Interactions

Published:1996-01-01 Issue:18 Volume:39 Page:3491-3502
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hedberg Martin H.¹,Jansen Johanna M.¹,Nordvall Gunnar¹,Hjorth Stephan¹,Unelius Lena¹,Johansson Anette M.¹

Affiliation:

1. Organic Pharmaceutical Chemistry, Uppsala University, Uppsala Biomedical Centre, Box 574, S-751 23 Uppsala, Sweden, Preclinical R&D, Astra Arcus AB, S-151 85 Södertälje, Sweden, and Department of Pharmacology, University of Göteborg, Medicinaregatan 7, S-413 90 Göteborg, Sweden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960188q

Reference73 articles.

1. Synthesis, structure, and antiparasitic activity of sulfamoyl derivatives of ribavirin

2. Aporphines as antagonists of dopamine D-1 receptors

3. Long-acting dihydropyridine calcium antagonists. 5. Synthesis and structure-activity relationships for a series of 2-[[(N-substituted-heterocyclyl)ethoxy]methyl]-1,4-dihydropyridine calcium antagonists

4. (R)-(-)-10-Methyl-11-hydroxyaporphine: a highly selective serotonergic agonist

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