Dimerization Inhibitors of HIV-1 Protease Based on a Bicyclic Guanidinium Subunit-Reference-Cited by-同舟云学术

Dimerization Inhibitors of HIV-1 Protease Based on a Bicyclic Guanidinium Subunit

Published:2003-10-23 Issue:24 Volume:46 Page:5196-5207
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Breccia Perla¹,Boggetto Nicole¹,Pérez-Fernández Ruth¹,Van Gool Michiel¹,Takahashi Masayuki¹,René Loïc¹,Prados Pilar¹,Badet Bernard¹,Reboud-Ravaux Michèle¹,de Mendoza Javier¹

Affiliation:

1. Departamento de Química Orgánica, Universidad Autónoma de Madrid, Cantoblanco, 28049 Madrid, Spain, Institut Jacques Monod, CNRS-Université Paris 6 & 7, 2, Place Jussieu-Tour 43, 75251 Paris Cedex 05, France, FRE2230 CNRS & Université de Nantes, F-44322 Nantes Cedex 3, France, and Institut de Chimie des Substances Naturelles-UPRS 2301 CNRS, 91198 Gif-sur-Yvette Cedex, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030871u

Reference30 articles.

1. The HIV-1 Protease as a Therapeutic Target for AIDS

2. Conserved Folding in Retroviral Proteases: Crystal Structure of Synthetic HIV-1 Protease

3. A structural model for the retroviral proteases

4. Mechanisms of HIV-1 drug resistance

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