Potent, Selective, Orally Active 3-Oxo-1,4-benzodiazepine GPIIb/IIIa Integrin Antagonists-Reference-Cited by-同舟云学术

Potent, Selective, Orally Active 3-Oxo-1,4-benzodiazepine GPIIb/IIIa Integrin Antagonists

Published:1996-01-01 Issue:25 Volume:39 Page:4867-4870
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Samanen James M.¹,Ali Fadia E.¹,Barton Linda S.¹,Bondinell William E.¹,Burgess Joelle L.¹,Callahan James F.¹,Calvo Raul R.¹,Chen Wenting¹,Chen Lichong¹,Erhard Karl¹,Feuerstein Giora¹,Heys Richard¹,Hwang Shing-Mei¹,Jakas Dalia R.¹,Keenan Richard M.¹,Ku Thomas W.¹,Kwon Chet¹,Lee Chao-Pin¹,Miller William H.¹,Newlander Kenneth A.¹,Nichols Andrew¹,Parker Michael¹,Peishoff Catherine E.¹,Rhodes Gerald¹,Ross Steven¹,Shu Arthur¹,Simpson Richard¹,Takata Dennis¹,Yellin Tobias O.¹,Uzsinskas Irene¹,Venslavsky Joseph W.¹,Yuan Chuan-Kui¹,Huffman William F.¹

Affiliation:

1. Department of Medicinal Chemistry, Radiochemistry Department, Department of Cellular Biochemistry, Pharmaceutical Sciences, Pharmacology Department, Department of Physical/Structural Chemistry, and Department of Pharmacokinetics, SmithKline Beecham Pharmaceuticals, King of Prussia, Pennsylvania 19406

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960558a

Reference18 articles.

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2. Nichols, A. J.; Vasko, J. A.; Koster, P. F.; Valocik, R. E.; Samanen, J. M. GPIIb/IIIa Antagonists as Novel Antithrombotic Drugs: Potential Therapeutic Agents. InCellular Adhesion: Molecular Definition to Therapeutic Potential; Metcalf, B. W., Dalton, B. J., Poste, G., Eds.; Plenum Press: New York, 1994; pp 213−237.

3. Lipid Particles May Help Solve Puzzle Regarding Genesis of Some Cardiovascular Diseases

4. Conformations of Arg-Gly-Asp containing heterodetic cyclic peptides: solution and crystal studies

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