Importance of Gastric Secretion and the Rapid Gastric Emptying of Ingested Water along the Lesser Curvature (“Magenstraße”) in Predicting the In Vivo Performance of Liquid Oral Dosage Forms in the Fed State Using a Modeling and Simulation-Reference-Cited by-同舟云学术

Importance of Gastric Secretion and the Rapid Gastric Emptying of Ingested Water along the Lesser Curvature (“Magenstraße”) in Predicting the In Vivo Performance of Liquid Oral Dosage Forms in the Fed State Using a Modeling and Simulation

Published:2022-01-25 Issue:2 Volume:19 Page:642-653
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Kiyota Tsuyoshi¹,Kambayashi Atsushi¹²^ORCID,Takagi Toshihide³^ORCID,Yamashita Shinji³^ORCID

Affiliation:

1. Pharmaceutical Research and Technology Labs, Astellas Pharma Inc., 180 Ozumi, Yaizu, Shizuoka 425-0072, Japan

2. School of Pharmaceutical Sciences, University of Shizuoka, 52-1 Yada, Suruga-ku, Shizuoka 422-8526, Japan

3. Faculty of Pharmaceutical Sciences, Setsunan University, 45-1 Nagaotoge-cho, Hirakata, Osaka 573-0101, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.molpharmaceut.1c00778

Reference50 articles.

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3. US Food and Drug Administration. Guidance for Industry: Food-Effect Bioavailability and Fed Bioequivalence Studies, 2002.

4. US Food and Drug Administration. Guidance for Industry: Assessing the Effects of Food on Drugs in INDs and NDAs (Draft Guidance), 2019.

5. European Medicines Agency. Guideline on the Investigation of Drug Interactions, 2012, (CPMP/EWP/560/95/Rev. 1).

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