Molecular Docking-Based Design and Development of a Highly Selective Probe Substrate for UDP-glucuronosyltransferase 1A10-Reference-Cited by-同舟云学术

Molecular Docking-Based Design and Development of a Highly Selective Probe Substrate for UDP-glucuronosyltransferase 1A10

Published:2018-02-08 Issue:3 Volume:15 Page:923-933
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Juvonen Risto O.¹^ORCID,Rauhamäki Sanna,Kortet Sami,Niinivehmas Sanna,Troberg Johanna²,Petsalo Aleksanteri¹,Huuskonen Juhani,Raunio Hannu¹,Finel Moshe²^ORCID,Pentikäinen Olli T.³^ORCID

Affiliation:

1. School of Pharmacy, Faculty of Health Sciences, University of Eastern Finland, Box 1627, FI-70211 Kuopio, Finland

2. Division of Pharmaceutical Chemistry and Technology, Faculty of Pharmacy, University of Helsinki, P.O. Box 56, FI-00014 Helsinki, Finland

3. Institute of Biomedicine, Faculty of Medicine, University of Turku, FI-20014 Turku, Finland

Funder

Sigrid Jus?liuksen S??ti?

Suomen Akatemia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.molpharmaceut.7b00871

Reference45 articles.

1. Gut Wall Metabolism. Application of Pre-Clinical Models for the Prediction of Human Drug Absorption and First-Pass Elimination

2. Intestinal glucuronidation metabolism may have a greater impact on oral bioavailability than hepatic glucuronidation metabolism in humans: A study with raloxifene, substrate for UGT1A1, 1A8, 1A9, and 1A10

3. Intestinal UGTs as potential modifiers of pharmacokinetics and biological responses to drugs and xenobiotics

4. First-Pass Metabolism via UDP-Glucuronosyltransferase: a Barrier to Oral Bioavailability of Phenolics

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