Influence of Physiological Gastrointestinal Surfactant Ratio on the Equilibrium Solubility of BCS Class II Drugs Investigated Using a Four Component Mixture Design
Author:
Affiliation:
1. Strathclyde Institute of Pharmacy and Biomedical Sciences, University of Strathclyde, 161 Cathedral Street, Glasgow G4 0RE, United Kingdom
Funder
FP7 Health
Cancer Research UK
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Pharmaceutical Science,Molecular Medicine
Link
http://pubs.acs.org/doi/pdf/10.1021/acs.molpharmaceut.7b00354
Reference46 articles.
1. A review of drug solubility in human intestinal fluids: Implications for the prediction of oral absorption
2. Early pharmaceutical profiling to predict oral drug absorption: Current status and unmet needs
3. Composition and Physicochemical Properties of Fasted‐State Human Duodenal and Jejunal Fluid: A Critical Evaluation of the Available Data
4. Postprandial Changes in Solubilizing Capacity of Human Intestinal Fluids for BCS Class II Drugs
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