Imaging Bradykinin B1 Receptor with 68Ga-Labeled [des-Arg10]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake-Reference-Cited by-同舟云学术

Imaging Bradykinin B1 Receptor with 68Ga-Labeled [des-Arg10]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake

Published:2015-07-02 Issue:8 Volume:12 Page:2879-2888
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Amouroux Guillaume¹,Pan Jinhe¹,Jenni Silvia¹,Zhang Chengcheng¹,Zhang Zhengxing¹,Hundal-Jabal Navjit¹,Colpo Nadine¹,Liu Zhibo²,Bénard François¹³,Lin Kuo-Shyan¹³

Affiliation:

1. Department of Molecular Oncology, BC Cancer Agency, Vancouver, BC V5Z 1L3, Canada

2. Chemistry Department, University of British Columbia, Vancouver, BC V6T 1Z1, Canada

3. Department of Radiology, University of British Columbia, Vancouver, BC V5Z 4E3, Canada

Funder

Canadian Institutes of Health Research

Leading Edge Endowment Fund

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.molpharmaceut.5b00070

Reference52 articles.

1. Non-peptide antagonists for kinin B1 receptors: new insights into their therapeutic potential for the management of inflammation and pain

2. Kinin B1receptors: key G-protein-coupled receptors and their role in inflammatory and painful processes

3. International Union of Pharmacology. XLV. Classification of the Kinin Receptor Family: from Molecular Mechanisms to Pathophysiological Consequences

4. Transcription Factor Nuclear Factor κB Regulates the Inducible Expression of the Human B1 Receptor Gene in Inflammation

5. Stimulation of the bradykinin B1 receptor induces the proliferation of estrogen-sensitive breast cancer cells and activates the ERK1/2 signaling pathway

Cited by 22 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Assessment of Radiolabelled Derivatives of R954 for Detection of Bradykinin B1 Receptor in Cancer Cells: Studies on Glioblastoma Xenografts in Mice;Pharmaceuticals;2024-07-07

2. Synthesis and Evaluation of Novel 68Ga-Labeled [D-Phe6,Leu13ψThz14]bombesin(6-14) Analogs for Cancer Imaging with Positron Emission Tomography;Pharmaceuticals;2024-05-11

3. [212Pb]Pb-eSOMA-01: A Promising Radioligand for Targeted Alpha Therapy of Neuroendocrine Tumors;Pharmaceuticals;2023-07-10

4. 68Ga-Labeled [Thz14]Bombesin(7–14) Analogs: Promising GRPR-Targeting Agonist PET Tracers with Low Pancreas Uptake;Molecules;2023-02-20

5. 68Ga-Labeled [Leu13ψThz14]Bombesin(7–14) Derivatives: Promising GRPR-Targeting PET Tracers with Low Pancreas Uptake;Molecules;2022-06-11