Islatravir Case Study for Enhanced Screening of Thermodynamically Stable Crystalline Anhydrate Phases in Pharmaceutical Process Development by Hot Melt Extrusion-Reference-Cited by-同舟云学术

Islatravir Case Study for Enhanced Screening of Thermodynamically Stable Crystalline Anhydrate Phases in Pharmaceutical Process Development by Hot Melt Extrusion

Published:2020-06-08 Issue:8 Volume:17 Page:2874-2881
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Skomski Daniel¹^ORCID,Varsolona Richard J.¹,Su Yongchao²^ORCID,Zhang Jingtao³^ORCID,Teller Ryan²,Forster Seth P.²,Barrett Stephanie Elizabeth¹,Xu Wei²

Affiliation:

1. MRL, Merck & Co., Inc., 126 East Lincoln Avenue, Rahway, New Jersey 07065, United States

2. MRL, Merck & Co. Inc, 770 Sumneytown Pike, West Point, Pennsylvania 19486, United States

3. MRL, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, New Jersey 07033, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.molpharmaceut.0c00316

Reference18 articles.

1. Dealing with the Impact of Ritonavir Polymorphs on the Late Stages of Bulk Drug Process Development

2. Elucidation of crystal form diversity of the HIV protease inhibitor ritonavir by high-throughput crystallization

3. Manipulating Hydrate Formation During High Shear Wet Granulation Using Polymeric Excipients

4. Solvent-Mediated Phase Transformation Kinetics of an Anhydrate/Hydrate System

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