Grafting Aminocyclopentane Carboxylic Acids onto the RGD Tripeptide Sequence Generates Low Nanomolar αVβ3/αVβ5 Integrin Dual Binders-Reference-Cited by-同舟云学术

Grafting Aminocyclopentane Carboxylic Acids onto the RGD Tripeptide Sequence Generates Low Nanomolar αVβ3/αVβ5 Integrin Dual Binders

Published:2005-11-04 Issue:24 Volume:48 Page:7675-7687
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Casiraghi Giovanni¹,Rassu Gloria¹,Auzzas Luciana¹,Burreddu Paola¹,Gaetani Enrico¹,Battistini Lucia¹,Zanardi Franca¹,Curti Claudio¹,Nicastro Giuseppe¹,Belvisi Laura¹,Motto Ilaria¹,Castorina Massimo¹,Giannini Giuseppe¹,Pisano Claudio¹

Affiliation:

1. Dipartimento Farmaceutico, Università di Parma, Parco Area delle Scienze 27A, I-43100 Parma, Italy, Istituto di Chimica Biomolecolare del CNR, Traversa La Crucca 3, I-07040 Li Punti, Sassari, Italy, Centro Interfacoltà Misure “G. Casnati”, Università di Parma, Parco Area delle Scienze 23A, I-43100 Parma, Italy, Dipartimento di Chimica Organica e Industriale, Università di Milano, Via Venezian 21, I-20133 Milano, Italy, and Sigma-Tau, Research & Development, Via Pontina Km 30.400, 00040 Pomezia, Roma, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm050698x

Reference60 articles.

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