New β-Alanine Derivatives Are Orally Available Glucagon Receptor Antagonists-Reference-Cited by-同舟云学术

New β-Alanine Derivatives Are Orally Available Glucagon Receptor Antagonists

Published:2007-01-01 Issue:1 Volume:50 Page:113-128
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Lau Jesper¹,Behrens Carsten¹,Sidelmann Ulla G.¹,Knudsen Lotte B.¹,Lundt Behrend¹,Sams Christian¹,Ynddal Lars¹,Brand Christian L.¹,Pridal Lone¹,Ling Anthony¹,Kiel Dan¹,Plewe Michael¹,Shi Shengua¹,Madsen Peter¹

Affiliation:

1. Protein Engineering, Discovery Biology Management, Medicinal Chemistry, Insulin Engineering, Drug Metabolism, Pharmacology Research, and Screening & Assay Technology, Novo Nordisk A/S, Novo Nordisk Park, DK-2760 Måløv, Denmark, and Departments of Medicinal Chemistry, Computational Chemistry, and Pharmacology, Pfizer Global Research and Development, 10770 Science Center Drive, San Diego, California 92121

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm058026u

Reference32 articles.

1. Introduction

2. Predominant Role of Gluconeogenesis in Increased Hepatic Glucose Production in NIDDM

3. Glucagon: Role in the Hyperglycemia of Diabetes Mellitus

4. Prevention of Human Diabetic Ketoacidosis by Somatostatin

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