Enthalpic Efficiency of Ligand Binding
Author:
Affiliation:
1. Sanofi-Aventis CHINOIN, 1−5. Tó u, Budapest, Hungary, H-1045, and Discovery Chemistry, Gedeon Richter Plc., 19−21. Gyõmrői út, Budapest, Hungary, H-1103
Publisher
American Chemical Society (ACS)
Subject
Library and Information Sciences,Computer Science Applications,General Chemical Engineering,General Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/ci100125a
Reference28 articles.
1. The maximal affinity of ligands
2. The role of molecular size in ligand efficiency
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4. Ligand efficiency: a useful metric for lead selection
5. Ligand efficiency indices as guideposts for drug discovery
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