Total Synthesis of LFA-1 Antagonist BIRT-377 via Organocatalytic Asymmetric Construction of a Quaternary Stereocenter-Reference-Cited by-同舟云学术

Total Synthesis of LFA-1 Antagonist BIRT-377 via Organocatalytic Asymmetric Construction of a Quaternary Stereocenter

Published:2005-01-28 Issue:5 Volume:7 Page:867-870
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Chowdari Naidu S.¹,Barbas Carlos F.¹

Affiliation:

1. The Skaggs Institute for Chemical Biology and the Departments of Chemistry and Molecular Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ol047368b

Reference71 articles.

1. Self-Regeneration of Stereocenters: A Practical Enantiospecific Synthesis of LFA-1 Antagonist BIRT-377

2. An Improved Synthesis of Chiral α-(4-Bromobenzyl)alanine Ethyl Ester and Its Application to the Synthesis of LFA-1 Antagonist BIRT-377

3. (c) Stehle, S.; Nummy, L.; Yee, N.Tetrahedron: Asymmetry2001,12, 101.

4. Crystallization-induced asymmetric transformations and self-regeneration of stereocenters (SROSC): enantiospecific synthesis of α-benzylalanine and hydantoin BIRT-377

5. (e) Yee, N.; Nummy, L. J.; Frutos, R. P.; Song, J. J.; Napolitano, E.; Byrne, D. P.; Jones, P. J.; Farina, V.Tetrahedron: Asymmetry2003,14, 3495.

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