Synthesis and Biological Activity of NK-1 Selective, N-Backbone Cyclic Analogs of the C-Terminal Hexapeptide of Substance P
Author:
Affiliation:
1. Departments of Organic Chemistry and Biological Chemistry, The Hebrew University of Jerusalem, Jerusalem 91904, Israel
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm960154i
Reference27 articles.
1. Neurokinin B is a preferred agonist for a neuronal substance P receptor and its action is antagonized by enkephalin.
2. Highly selective agonists for substance P receptor subtypes.
3. Characterization of a neurokinin B receptor site in rat brain using a highly selective radioligand.
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