Identification of a Novel Series of Orexin Receptor Antagonists with a Distinct Effect on Sleep Architecture for the Treatment of Insomnia
Author:
Affiliation:
1. Medicinal Chemistry, Aurigene Discovery Technologies, 39-40, Electronic City Phase 2, Bangalore 560 100, India
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm4007627
Reference56 articles.
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2. The hypocretins: Hypothalamus-specific peptides with neuroexcitatory activity
3. Physiology of the orexinergic/hypocretinergic system: a revisit in 2012
4. Central functions of the orexinergic system
5. Orexin/Hypocretin: A Neuropeptide at the Interface of Sleep, Energy Homeostasis, and Reward System
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