Syntheses and Opioid Receptor Binding Affinities of 8-Amino-2,6-methano-3-benzazocines-Reference-Cited by-同舟云学术

Syntheses and Opioid Receptor Binding Affinities of 8-Amino-2,6-methano-3-benzazocines

Published:2003-02-01 Issue:5 Volume:46 Page:838-849
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wentland Mark P.¹,Ye Yingchun¹,Cioffi Christopher L.¹,Lou Rongliang¹,Zhou Qun¹,Xu Guoyou¹,Duan Wenhu¹,Dehnhardt Christoph M.¹,Sun Xufeng¹,Cohen Dana J.¹,Bidlack Jean M.¹

Affiliation:

1. Department of Chemistry, Rensselaer Polytechnic Institute, Troy, New York 12180, and Department of Pharmacology and Physiology, School of Medicine and Dentistry, University of Rochester, Rochester, New York 14642

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020429w

Reference55 articles.

1. Cyclazocine revisited

2. (+)-cis-N-(para-, meta-, and ortho-substituted benzyl)-N-normetazocines: Synthesis and binding affinity at the [3H]-(+)-pentazocine-labeled (.sigma.1) site and quantitative structure-affinity relationship studies

3. Deoxymorphines: role of the phenolic hydroxyl in antinociception and opiate receptor interactions

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