Identification and Characterization of Small Molecule Inhibitors of a Class I Histone Deacetylase from Plasmodium falciparum-Reference-Cited by-同舟云学术

Identification and Characterization of Small Molecule Inhibitors of a Class I Histone Deacetylase from Plasmodium falciparum

Published:2009-03-24 Issue:8 Volume:52 Page:2185-2187
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Patel Vishal¹,Mazitschek Ralph¹,Coleman Bradley¹,Nguyen Cokey¹,Urgaonkar Sameer¹,Cortese Joseph¹,Barker Robert H.¹,Greenberg Edward¹,Tang Weiping¹,Bradner James E.¹,Schreiber Stuart L.¹,Duraisingh Manoj T.¹,Wirth Dyann F.¹,Clardy Jon¹

Affiliation:

1. Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, Boston, Massachusetts, Department of Immunology and Infectious Disease, Harvard School of Public Health, Boston, Massachusetts, Broad Institute of Massachusetts Institute of Technology and Harvard University, Cambridge, Massachusetts, and Genzyme Corporation, Framingham, Massachusetts

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm801654y

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2. Resistance mutations reveal the atovaquone-binding domain of cytochrome b in malaria parasites

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5. Chromatin Modifications and Their Function

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