Discovery of EGFR Selective 4,6-Disubstituted Pyrimidines from a Combinatorial Kinase-Directed Heterocycle Library-Reference-Cited by-同舟云学术

Discovery of EGFR Selective 4,6-Disubstituted Pyrimidines from a Combinatorial Kinase-Directed Heterocycle Library

Published:2006-01-31 Issue:7 Volume:128 Page:2182-2183
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Zhang Qiong¹,Liu Yi¹,Gao Feng¹,Ding Qiang¹,Cho Charles¹,Hur Wooyoung¹,Jin Yunho¹,Uno Tetsuo¹,Joazeiro Claudio A. P.¹,Gray Nathanael¹

Affiliation:

1. Departments of Chemistry and Cell Biology, Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, and Department of Chemistry, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja0567485

Reference14 articles.

1. Chemogenomics: an emerging strategy for rapid target and drug discovery

2. EGFRMutation and Resistance of Non–Small-Cell Lung Cancer to Gefitinib

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