Nonsymmetric P2/P2‘ Cyclic Urea HIV Protease Inhibitors. Structure−Activity Relationship, Bioavailability, and Resistance Profile of Monoindazole-Substituted P2 Analogues-Reference-Cited by-同舟云学术

Nonsymmetric P2/P2‘ Cyclic Urea HIV Protease Inhibitors. Structure−Activity Relationship, Bioavailability, and Resistance Profile of Monoindazole-Substituted P2 Analogues

Published:1998-06-01 Issue:13 Volume:41 Page:2411-2423
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

De Lucca George V.¹,Kim Ui T.¹,Liang Jing¹,Cordova Beverly¹,Klabe Ronald M.¹,Garber Sena¹,Bacheler Lee T.¹,Lam Gilbert N.¹,Wright Matthew R.¹,Logue Kelly A.¹,Erickson-Viitanen Susan¹,Ko Soo S.¹,Trainor George L.¹

Affiliation:

1. Dupont Merck Pharmaceutical Company, Experimental Station, P.O. Box 80500, Wilmington, Delaware 19880-0500

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm980103g

Reference34 articles.

1. Update on a proteinase inhibitor

2. L-735,524: an orally bioavailable human immunodeficiency virus type 1 protease inhibitor.

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