Development of Potent and Selective Inhibitors of Aldo–Keto Reductase 1C3 (Type 5 17β-Hydroxysteroid Dehydrogenase) Based on N-Phenyl-Aminobenzoates and Their Structure–Activity Relationships-Reference-Cited by-同舟云学术

Development of Potent and Selective Inhibitors of Aldo–Keto Reductase 1C3 (Type 5 17β-Hydroxysteroid Dehydrogenase) Based on N-Phenyl-Aminobenzoates and Their Structure–Activity Relationships

Published:2012-02-15 Issue:5 Volume:55 Page:2311-2323
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Adeniji Adegoke O.¹,Twenter Barry M.²,Byrns Michael C.¹,Jin Yi¹,Chen Mo¹,Winkler Jeffrey D.²,Penning Trevor M.¹

Affiliation:

1. Department of Pharmacology and Center of Excellence in Environmental Toxicology, Perelman School of Medicine, University of Pennsylvania, 130C John Morgan Building, 3620 Hamilton Walk, Philadelphia, Pennsylvania 19104-6084, United States

2. Department of Chemistry, University of Pennsylvania, 231 South 34th Street, Philadelphia, Pennsylvania 19104, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201547v

Reference52 articles.

1. Cancer Statistics, 2010

2. Partners in crime: deregulation of AR activity and androgen synthesis in prostate cancer

3. Starving the Addiction: New Opportunities for Durable Suppression of AR Signaling in Prostate Cancer

4. Androgen Levels Increase by IntratumoralDe novoSteroidogenesis during Progression of Castration-Resistant Prostate Cancer

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