Development of a Conformational Histamine H3 Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists-Reference-Cited by-同舟云学术

Development of a Conformational Histamine H3 Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists

Published:2020-05-13 Issue:6 Volume:5 Page:1734-1742
ISSN:2379-3694
Container-title:ACS Sensors
language:en
Short-container-title:ACS Sens.

Author:

Schihada Hannes¹²^ORCID,Ma Xiaoyuan³,Zabel Ulrike²,Vischer Henry F.³^ORCID,Schulte Gunnar¹^ORCID,Leurs Rob³^ORCID,Pockes Steffen⁴,Lohse Martin J.²⁵⁶

Affiliation:

1. Section of Receptor Biology & Signaling, Dept. Physiology & Pharmacology, Karolinska Institutet, Stockholm 171 77, Sweden

2. Institute of Pharmacology and Toxicology and Rudolf Virchow Center, University of Würzburg, Würzburg 97070, Germany

3. Amsterdam Institute for Molecules, Medicines and Systems, Division of Medicinal Chemistry, Faculty of Science, Vrije Universiteit Amsterdam, Amsterdam 1081 HV, The Netherlands

4. Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Regensburg 93053, Germany

5. ISAR Bioscience, Planegg 82152, Germany

6. Max Delbrück Center for Molecular Medicine, Berlin 13125, Germany

Funder

Bundesministerium für Bildung und Forschung

Vetenskapsrådet

Deutsche Forschungsgemeinschaft

China Scholarship Council

Cancerfonden

Karolinska Institutet

National Institutes of Health

Publisher

American Chemical Society (ACS)

Subject

Fluid Flow and Transfer Processes,Process Chemistry and Technology,Instrumentation,Bioengineering

Link

http://pubs.acs.org/doi/pdf/10.1021/acssensors.0c00397

Reference38 articles.

1. International Union of Basic and Clinical Pharmacology. XCVIII. Histamine Receptors

2. Evaluation of the CNS properties of SCH 29851, a potential non-sedating antihistamine

3. Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

4. The Histamine H3 Receptor: Structure, Pharmacology, and Function

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