A Novel Selective GABAA α1 Receptor Agonist Displaying Sedative and Anxiolytic-like Properties in Rodents-Reference-Cited by-同舟云学术

A Novel Selective GABAA α1 Receptor Agonist Displaying Sedative and Anxiolytic-like Properties in Rodents

Published:2005-09-23 Issue:21 Volume:48 Page:6756-6760
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Selleri Silvia¹,Bruni Fabrizio¹,Costagli Camilla¹,Costanzo Annarella¹,Guerrini Gabriella¹,Ciciani Giovanna¹,Gratteri Paola¹,Besnard François¹,Costa Barbara¹,Montali Marina¹,Martini Claudia¹,Fohlin Jonna¹,De Siena Gaetano¹,Aiello Petra Malmberg¹

Affiliation:

1. Department of Pharmaceutical Sciences, University of Firenze, Via U. Schiff 6, 50019 Sesto Fiorentino, Italy, Department of Molecular and Functional Genomics, Synthélabo, 10 rue des Carrîeres, 92500 Rueil-Malmaison, France, Department of Psychiatry, Neurobiology, Pharmacology e Biotechnologies, University of Pisa, Via Bonanno 6, 56126 Pisa, Italy, and Department of Preclinical and Clinical Pharmacology, University of Firenze, Viale Pieraccini 6, 50139 Firenze, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm058002n

Reference21 articles.

1. Subunit Composition, Distribution and Function of GABA-A Receptor Subtypes

2. Specific GABAA circuits in brain development and therapy

3. Different types of GABA A receptors may mediate the anticonflict and response rate-decreasing effects of zaleplon, zolpidem, and midazolam in squirrel monkeys

4. Anxioselective anxiolytics: can less be more?

5. β-CCT, a selective BZ-ω1 receptor antagonist, blocks the anti-anxiety but not the amnesic action of chlordiazepoxide in mice

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