Michael Acceptor Based Antiplasmodial and Antitrypanosomal Cysteine Protease Inhibitors with Unusual Amino Acids-Reference-Cited by-同舟云学术

Michael Acceptor Based Antiplasmodial and Antitrypanosomal Cysteine Protease Inhibitors with Unusual Amino Acids

Published:2010-02-04 Issue:5 Volume:53 Page:1951-1963
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Breuning Alexander¹,Degel Björn¹,Schulz Franziska¹,Büchold Christian¹,Stempka Martin¹²,Machon Uwe³,Heppner Saskia⁴,Gelhaus Christoph⁴,Leippe Matthias⁴,Leyh Matthias²,Kisker Caroline²,Rath Jennifer⁵,Stich August⁵,Gut Jiri⁶,Rosenthal Philip J.⁶,Schmuck Carsten³,Schirmeister Tanja¹

Affiliation:

1. Institute of Pharmacy and Food Chemistry, University of Würzburg, Am Hubland, 97074 Würzburg, Germany

2. Rudolf-Virchow-Zentrum, DFG-Forschungszentrum für Experimentelle Biomedizin, University of Würzburg, Josef-Schneider-Strasse 2, 97080 Würzburg, Germany

3. Institute of Organic Chemistry, University of Duisburg-Essen, Universitätstrasse 7, 45141 Essen, Germany

4. Institute of Zoology, University of Kiel, Olshausenstrasse 40, 24098 Kiel, Germany

5. Department of Tropical Medicine, Medical Mission Institute, Salvatorstrasse 7, 97074 Würzburg, Germany

6. Department of Medicine, San Francisco General Hospital, University of California, San Francisco, Box 0811, San Francisco, California 94143

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm900946n

Reference45 articles.

1. Human African trypanosomiasis: clinical presentation and immune response

2. Cysteine Proteinases of Trypanosome Parasites Novel Targets for Chemotherapy

3. Chemotherapeutic Agents Against Malaria: What Next After Chloroquine?

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