Solid-Phase Synthesis of Tetrahydro-1,4-benzodiazepine-2-one Derivatives as a β-Turn Peptidomimetic Library-Reference-Cited by-同舟云学术

Solid-Phase Synthesis of Tetrahydro-1,4-benzodiazepine-2-one Derivatives as a β-Turn Peptidomimetic Library

Published:2004-01-08 Issue:2 Volume:6 Page:207-213
ISSN:1520-4766
Container-title:Journal of Combinatorial Chemistry
language:en
Short-container-title:J. Comb. Chem.

Author:

Im Isak¹,Webb Thomas R.¹,Gong Young-Dae¹,Kim Jae-Il¹,Kim Yong-Chul¹

Affiliation:

1. Department of Life Science, Kwangju Institute of Science and Technology, Gwangju 500-712, Republic of Korea, ChemBridge Research Labs, LLC, and ChemBridge Corporation, San Diego, California 92127, and Medicinal Science Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea

Publisher

American Chemical Society (ACS)

Subject

General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cc034039m

Reference29 articles.

1. Converting a Peptide into a Drug: Strategies to Improve Stability and Bioavailability

2. Identification of a Potent Heterocyclic Ligand To Somatostatin Receptor Subtype 5 by the Synthesis and Screening of β-Turn Mimetic Libraries

3. Synthesis and evaluation of a library of peptidomimetics based upon the β-turn

4. Expedient solid-phase synthesis of putative β-turn mimetics incorporating the i + 1, i + 2, and i + 3 sidechains

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