Design, Synthesis, and Preliminary Pharmacological Evaluation of a Set of Small Molecules That Directly Activate Gi Proteins-Reference-Cited by-同舟云学术

Design, Synthesis, and Preliminary Pharmacological Evaluation of a Set of Small Molecules That Directly Activate Gi Proteins

Published:2005-09-10 Issue:20 Volume:48 Page:6491-6503
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Manetti Dina¹,Di Cesare Mannelli Lorenzo¹,Dei Silvia¹,Galeotti Nicoletta¹,Ghelardini Carla¹,Romanelli Maria Novella¹,Scapecchi Serena¹,Teodori Elisabetta¹,Pacini Alessandra¹,Bartolini Alessandro¹,Gualtieri Fulvio¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Università di Firenze, Via U. Schiff 6, I-50019 Sesto Fiorentino (FI), Italy; Dipartimento di Farmacologia Preclinica e Clinica, Università di Firenze, Viale G. Pieraccini 6, I-50139 Firenze, Italy; and Dipartimento di Anatomia, Istologia e Medicina Legale, Università di Firenze, Viale G. Morgagni 85, I-50134 Firenze, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm050498l

Reference58 articles.

1. G protein antagonists

2. Regulators of G-protein signalling: a novel protein family involved in timely deactivation and desensitization of signalling via heterotrimeric G proteins

3. Activation of Heterotrimeric G-protein Signaling by a Ras-related Protein

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