Molecular Determinants of EphA2 and EphB2 Antagonism Enable the Design of Ligands with Improved Selectivity-Reference-Cited by-同舟云学术

Molecular Determinants of EphA2 and EphB2 Antagonism Enable the Design of Ligands with Improved Selectivity

Published:2023-11-01 Issue:21 Volume:63 Page:6900-6911
ISSN:1549-9596
Container-title:Journal of Chemical Information and Modeling
language:en
Short-container-title:J. Chem. Inf. Model.

Author:

Guidetti Lorenzo¹^ORCID,Zappia Alfonso¹,Scalvini Laura¹^ORCID,Ferrari Francesca Romana¹,Giorgio Carmine¹,Castelli Riccardo¹^ORCID,Galvani Francesca¹^ORCID,Vacondio Federica¹^ORCID,Rivara Silvia¹^ORCID,Mor Marco¹²^ORCID,Urbinati Chiara³,Rusnati Marco³,Tognolini Massimiliano¹,Lodola Alessio¹^ORCID

Affiliation:

1. Dipartimento di Scienze degli Alimenti e del Farmaco, Università degli Studi di Parma, Parco Area delle Scienze 27/A, I- 43124 Parma, Italy

2. Microbiome Research Hub, Università degli Studi di Parma, Parco Area delle scienze 11/A, I- 43124 Parma, Italy

3. Dipartimento di Medicina Molecolare Traslazionale, Università degli Studi di Brescia, Brescia 25121, Italy

Funder

Associazione Italiana per la Ricerca sul Cancro

Regione Emilia-Romagna

Publisher

American Chemical Society (ACS)

Subject

Library and Information Sciences,Computer Science Applications,General Chemical Engineering,General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jcim.3c01064

Reference60 articles.

1. Cell–cell signaling via Eph receptors and ephrins

2. Ephrins and their Receptors: Binding versus Biology

3. Eph receptors and ephrins in cancer: bidirectional signalling and beyond

4. Eph-Ephrin Bidirectional Signaling in Physiology and Disease

5. Emerging strategies for EphA2 receptor targeting for cancer therapeutics

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