The Physicochemical Properties, in Vitro Metabolism and Pharmacokinetics of a Novel Ester Prodrug of EXP3174-Reference-Cited by-同舟云学术

The Physicochemical Properties, in Vitro Metabolism and Pharmacokinetics of a Novel Ester Prodrug of EXP3174

Published:2010-10-01 Issue:6 Volume:7 Page:2132-2140
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Yan Yi-Dong¹,Kim Han-Kyung¹,Seo Ki-Heon¹,Lee Won Seok¹,Lee Gwan-Sun¹,Woo Jong-Soo¹,Yong Chul-Soon¹,Choi Han-Gon¹

Affiliation:

1. College of Pharmacy, Yeungnam University, 214-1 Dae-Dong, Gyongsan 712-749, South Korea, Hanmi Research Centre, Hanmi Pharm Co. Ltd., Dongtam-myeon, 377-1 Hwaseong-si, Gyeonggi-do, 445-913, South Korea, and College of Pharmacy, Hanyang University, 1271, Sa-3-Dong, Ansan 426-791, South Korea

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/mp100166c

Reference29 articles.

1. Losartan Potassium

2. Pharmacokinetics of losartan, an angiotensin II receptor antagonist, and its active metabolite EXP3174 in humans

3. EXP3174: The Major Active Metabolite of Losartan

4. Angiotensin II Type 1 Receptor Blockers

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