Discovery of 3-{5-[(6-Amino-1H-pyrazolo[3,4-b]pyridine-3-yl)methoxy]-2-chlorophenoxy}-5-chlorobenzonitrile (MK-4965): A Potent, Orally Bioavailable HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitor with Improved Potency against Key Mutant Viruses-Reference-Cited by-同舟云学术

Discovery of 3-{5-[(6-Amino-1H-pyrazolo[3,4-b]pyridine-3-yl)methoxy]-2-chlorophenoxy}-5-chlorobenzonitrile (MK-4965): A Potent, Orally Bioavailable HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitor with Improved Potency against Key Mutant Viruses

Published:2008-10-23 Issue:20 Volume:51 Page:6503-6511
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tucker Thomas J.,Sisko John T.,Tynebor Robert M.,Williams Theresa M.,Felock Peter J.,Flynn Jessica A.,Lai Ming-Tain,Liang Yuexia,McGaughey Georgia,Liu Meiquing,Miller Mike,Moyer Gregory,Munshi Vandna,Perlow-Poehnelt Rebecca,Prasad Sridhar,Reid John C.,Sanchez Rosa,Torrent Maricel,Vacca Joseph P.,Wan Bang-Lin,Yan Youwei

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800856c

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