3-(4-Fluoropiperidin-3-yl)-2-phenylindoles as High Affinity, Selective, and Orally Bioavailable h5-HT2A Receptor Antagonists-Reference-Cited by-同舟云学术

3-(4-Fluoropiperidin-3-yl)-2-phenylindoles as High Affinity, Selective, and Orally Bioavailable h5-HT2A Receptor Antagonists

Published:2001-04-03 Issue:10 Volume:44 Page:1603-1614
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rowley Michael¹,Hallett David J.¹,Goodacre Simon¹,Moyes Christopher¹,Crawforth James¹,Sparey Timothy J.¹,Patel Smita¹,Marwood Rose¹,Patel Shil¹,Thomas Steven¹,Hitzel Laure¹,O'Connor Desmond¹,Szeto Nicola¹,Castro Jose L.¹,Hutson Peter H.¹,MacLeod Angus M.¹

Affiliation:

1. Merck Sharp and Dohme, The Neuroscience Research Centre, Terlings Park, Eastwick Road, Harlow, Essex CM20 2QR, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0004998

Reference28 articles.

1. Antipsychotic Drugs: Direct Correlation Between Clinical Potency and Presynaptic Action on Dopamine Neurons

2. A Clinical Guide to Antipsychotic Drugs

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