Access to Artemisinin–Triazole Antimalarials via Organo-Click Reaction: High In Vitro/In Vivo Activity against Multi-Drug-Resistant Malaria Parasites

Author:

Herrmann Lars1,Leidenberger Maria2,Quadros Helenita C.3ORCID,Grau Benedikt W.1,Hampel Frank1,Friedrich Oliver2,Moreira Diogo R. M.3ORCID,Kappes Barbara2,Tsogoeva Svetlana B.1ORCID

Affiliation:

1. Department of Chemistry and Pharmacy, Organic Chemistry Chair I and Interdisciplinary Center for Molecular Materials (ICMM), Friedrich-Alexander-University Erlangen-Nürnberg, Nikolaus Fiebiger-Straße 10, 91058 Erlangen, Germany

2. Institute of Medical Biotechnology, Friedrich-Alexander-University Erlangen-Nürnberg, Paul-Gordon-Straße 3, 91052 Erlangen, Germany

3. Fiocruz, Instituto Gonçalo Moniz, Salvador 40296-710, Bahia, Brazil

Funder

Funda??o Oswaldo Cruz

Funda??o de Amparo ? Pesquisa do Estado da Bahia

Deutsche Forschungsgemeinschaft

Conselho Nacional de Desenvolvimento Cient?fico e Tecnol?gico

Coordena??o de Aperfei?oamento de Pessoal de N?vel Superior

Publisher

American Chemical Society (ACS)

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