Exploring Polymorphism: Hydrochloride Salts of Pitolisant and Analogues-Reference-Cited by-同舟云学术

Exploring Polymorphism: Hydrochloride Salts of Pitolisant and Analogues

Published:2024-01-23 Issue: Volume: Page:
ISSN:1528-7483
Container-title:Crystal Growth & Design
language:en
Short-container-title:Crystal Growth & Design

Author:

Patel Jessica¹,Leduc Zachary¹,Nunez Avila Aaron Gabriel¹,Glover Joseph A.²,Wu Kelin³,Zhang Yuxing³,Zhang Jing³,Zhai Xiaoting³,Jing Huize³,Chen Alex M.³,Chartrand Daniel¹,Maris Thierry¹^ORCID,Day Graeme M.²^ORCID,Wuest James D.¹^ORCID

Affiliation:

1. Département de Chimie, Université de Montréal, Montréal, Québec H2V 0B3, Canada

2. School of Chemistry, University of Southampton, University Road, Southampton SO17 1BJ, United Kingdom

3. Crystal Pharmatech, B4-301, Biobay, 218 Xinghu Street, Suzhou Industrial Park, Suzhou 215123, China

Funder

Canada Foundation for Innovation

Canada Research Chairs

Natural Sciences and Engineering Research Council of Canada

H2020 European Research Council

Mitacs

Publisher

American Chemical Society (ACS)

Subject

Condensed Matter Physics,General Materials Science,General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.cgd.3c01245

Reference84 articles.

1. The histamine H3 receptor: from discovery to clinical trials with pitolisant

2. Raga, M.; Sallares, J.; Guerrero, M.; Guglietta, A.; Arrang, J.M.; Schwartz, J.C.; Stark, H.; Schunack, W.; Ligneau, X.; Lecomte, J.M.; Ganellin, C. Monohydrochloride Salt of 1-[3-[3-(4-Chlorophenyl)propoxy]propyl]piperidine. U.S. Patent US8,207,197 B2, 2012.

3. Raga, M.; Sallares, J.; Guerrero, M.; Guglietta, A. The Monohydrochloride Salt of 1-[3-[3-(4-Chlorophenyl)propoxy]propyl]piperidine. WO Patent WO2006/084833 A1, 2006.

4. Recent Advances in Polymorph Discovery Methods of Organic Crystals

5. Adding a Pinch of Salt: Using Ionic Mixed-Crystal Seeds to Search for New Solid Forms