A New Thermodynamically Favored Flubendazole/Maleic Acid Binary Crystal Form: Structure, Energetics, and in Silico PBPK Model-Based Investigation-Reference-Cited by-同舟云学术

A New Thermodynamically Favored Flubendazole/Maleic Acid Binary Crystal Form: Structure, Energetics, and in Silico PBPK Model-Based Investigation

Published:2018-02-27 Issue:4 Volume:18 Page:2377-2386
ISSN:1528-7483
Container-title:Crystal Growth & Design
language:en
Short-container-title:Crystal Growth & Design

Author:

de Araujo Gabriel L. B.^ORCID,Ferreira Fabio Furlan¹^ORCID,Bernardes Carlos E. S.²^ORCID,Sato Juliana A. P.¹,Gil Otávio M.,de Faria Dalva L. A.,Loebenberg Raimar³,Byrn Stephen R.,Ghisleni Daniela D. M.,Bou-Chacra Nadia A.,Pinto Terezinha J. A.,Antonio Selma G.⁴,Ferraz Humberto G.,Zemlyanov Dmitry,Gonçalves Débora S.,Minas da Piedade Manuel E.²

Affiliation:

1. Centro de Ciencias Naturais e Humanas, Universidade Federal do ABC (UFABC), Santo André, São Paulo, Brazil

2. Centro de Química e Bioquímica e Centro de Química Estrutural, Faculdade de Ciências, Universidade de Lisboa, 1748-016 Lisboa, Portugal

3. Faculty of Pharmacy & Pharmaceutical Sciences, University of Alberta, Edmonton, Alberta, Canada T6G 2H7

4. Departamento de Físico-Química, Instituto de Química, Universidade Estadual Paulista, Araraquara, Brazil

Funder

Conselho Nacional de Desenvolvimento Cient?fico e Tecnol?gico

Funda??o de Amparo ? Pesquisa do Estado de S?o Paulo

Funda??o para a Ci?ncia e a Tecnologia

Publisher

American Chemical Society (ACS)

Subject

Condensed Matter Physics,General Materials Science,General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.cgd.7b01807

Reference54 articles.

1. Flubendazole: a candidate macrofilaricide for lymphatic filariasis and onchocerciasis field programs

2. Effects of the benzimidazole anthelmintic drug flubendazole on rat embryos in vitro

3. Exploring the Potential of Flubendazole in Filariasis Control: Evaluation of the Systemic Exposure for Different Pharmaceutical Preparations

4. Progress and Impact of 13 Years of the Global Programme to Eliminate Lymphatic Filariasis on Reducing the Burden of Filarial Disease

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