5-HT1A- versus D2-Receptor Selectivity of Flesinoxan and Analogous N 4-Substituted N 1-Arylpiperazines-Reference-Cited by-同舟云学术

5-HT1A- versus D2-Receptor Selectivity of Flesinoxan and Analogous N 4-Substituted N 1-Arylpiperazines

Published:1997-01-01 Issue:3 Volume:40 Page:300-312
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kuipers Wilma¹,Kruse Chris G.¹,van Wijngaarden Ineke¹,Standaar Piet J.¹,Tulp Martin Th. M.¹,Veldman Nora¹,Spek Anthony L.¹,IJzerman Adriaan P.¹

Affiliation:

1. Departments of Medicinal Chemistry and CNS Pharmacology, Solvay Pharmaceuticals Research Laboratories, P.O. Box 900, 1380 DA Weesp, The Netherlands, Bijvoet Center for Biomolecular Research, Laboratory of Crystal and Structural Chemistry, Utrecht University, Padualaan 8, 3584 CH Utrecht, The Netherlands, and Division of Medicinal Chemistry, Leiden/Amsterdam Center for Drug Research, P.O. Box 9502, 2300 RA Leiden, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960496o

Reference49 articles.

1. 5-Hydroxytryptamine receptor subtypes in vertebrates and invertebrates

2. Serotonin Receptor Subtypes

3. 8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site

4. The concept of selectivity in 5-HT receptor research

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