Synthesis and Characterization of a BODIPY Conjugate of the BCR-ABL Kinase Inhibitor Tasigna (Nilotinib): Evidence for Transport of Tasigna and Its Fluorescent Derivative by ABC Drug Transporters-Reference-Cited by-同舟云学术

Synthesis and Characterization of a BODIPY Conjugate of the BCR-ABL Kinase Inhibitor Tasigna (Nilotinib): Evidence for Transport of Tasigna and Its Fluorescent Derivative by ABC Drug Transporters

Published:2011-06-16 Issue:4 Volume:8 Page:1292-1302
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Shukla Suneet¹,Skoumbourdis Amanda P.²,Walsh Martin J.²,Hartz Anika M. S.,Fung King Leung¹,Wu Chung-Pu¹,Gottesman Michael M.¹,Bauer Björn,Thomas Craig J.²,Ambudkar Suresh V.¹

Affiliation:

1. Laboratory of Cell Biology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892, United States

2. NIH Chemical Genomics Center, 9800 Medical Center Drive, Rockville, Maryland 20850, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/mp2001022

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