Potent and Selective Inhibitors of Platelet-Derived Growth Factor Receptor Phosphorylation. 1. Synthesis, Structure−Activity Relationship, and Biological Effects of a New Class of Quinazoline Derivatives-Reference-Cited by-同舟云学术

Potent and Selective Inhibitors of Platelet-Derived Growth Factor Receptor Phosphorylation. 1. Synthesis, Structure−Activity Relationship, and Biological Effects of a New Class of Quinazoline Derivatives

Published:2002-06-11 Issue:14 Volume:45 Page:3057-3066
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Matsuno Kenji¹,Ichimura Michio¹,Nakajima Takao¹,Tahara Keiko¹,Fujiwara Shigeki¹,Kase Hiroshi¹,Ushiki Junko¹,Giese Neill A.¹,Pandey Anjali¹,Scarborough Robert M.¹,Lokker Nathalie A.¹,Yu Jin-Chen¹,Irie Junko¹,Tsukuda Eiji¹,Ide Shin-ichi¹,Oda Shoji¹,Nomoto Yuji¹

Affiliation:

1. Pharmaceutical Research Institute, Kyowa Hakko Kogyo Company, Ltd., Shimotogari 1188, Nagaizumi-cho, Sunto-gun, Shizuoka 411-8731, Japan, and Millennium Pharmaceuticals, Inc., 256 East Grant Avenue, San Francisco, California 94108

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm010428o

Reference39 articles.

1. Mechanism of platelet-derived growth factor (PDGF) AA, AB, and BB binding to alpha and beta PDGF receptor.

2. Platelet-derived growth factor: Isoform-specific signalling via heterodimeric or homodimeric receptor complexes

3. Dimerization of extracellular domains of platelet-derived growth factor receptors. A revised model of receptor-ligand interaction

4. Signal transduction by receptors with tyrosine kinase activity

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