Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 1. Mapping the Central 5-HT3 Receptor Binding Site by Arylpiperazine Derivatives-Reference-Cited by-同舟云学术

Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 1. Mapping the Central 5-HT3 Receptor Binding Site by Arylpiperazine Derivatives

Published:1998-02-01 Issue:5 Volume:41 Page:728-741
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cappelli Andrea¹,Anzini Maurizio¹,Vomero Salvatore¹,Mennuni Laura¹,Makovec Francesco¹,Doucet Edith¹,Hamon Michel¹,Bruni Giancarlo¹,Romeo Maria R.¹,Menziani M. Cristina¹,De Benedetti Pier G.¹,Langer Thierry¹

Affiliation:

1. Dipartimento Farmaco Chimico Tecnologico, Università di Siena, Via Banchi di Sotto 55, 53100 Siena, Italy, Rotta Research Laboratorium S.p.A., Via Valosa di Sopra 7, 20052 Monza, Italy, Neurobiologie Cellulaire et Fonctionnelle, INSERM U288, Faculté de Médicine Pitié-Salpêtrière, 91, Boulevard de l'Hôpital, 75634 Paris Cedex 13, France, Istituto di Farmacologia, Università di Siena, Le Scotte 6, 53100 Siena, Italy, Dipartimento di Chimica, Università degli Studi di Modena, Via Campi 183, 41100 Modena,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970645i

Reference45 articles.

1. 5-HT3 receptors

2. Development of high-affinity 5-HT3 receptor antagonists. Structure-affinity relationships of novel 1,7-annulated indole derivatives. 1

3. The psychopharmacology of 5-HT3 receptors

4. Activation of a 5-HT3 receptor releases dopamine from rat striatal slice

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