Design of 2,5-Dimethyl-3-(6-dimethyl-4-methylpyridin-3-yl)-7-dipropylaminopyrazolo[1,5-a]pyrimidine (NBI 30775/R121919) and Structure−Activity Relationships of a Series of Potent and Orally Active Corticotropin-Releasing Factor Receptor Antagonists-Reference-Cited by-同舟云学术

Design of 2,5-Dimethyl-3-(6-dimethyl-4-methylpyridin-3-yl)-7-dipropylaminopyrazolo[1,5-a]pyrimidine (NBI 30775/R121919) and Structure−Activity Relationships of a Series of Potent and Orally Active Corticotropin-Releasing Factor Receptor Antagonists

Published:2004-08-06 Issue:19 Volume:47 Page:4787-4798
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Chen ¹,Wilcoxen Keith M.¹,Huang Charles Q.¹,Xie Yun-Feng¹,McCarthy James R.¹,Webb Thomas R.¹,Zhu Yun-Fei¹,Saunders John¹,Liu Xin-Jun¹,Chen Ta-Kung¹,Bozigian Haig¹,Grigoriadis Dimitri E.¹

Affiliation:

1. Neurocrine Biosciences, Inc., 10555 Sciences Center Drive, San Diego, California 92121

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm040058e

Reference58 articles.

1. Characterization of a 41-Residue Ovine Hypothalamic Peptide That Stimulates Secretion of Corticotropin and β-Endorphin

2. (b) De Souza, E. B.; Grigoriadis, D. E. InPsychopharmacology: The fourthgeneration of progress; Bloom, F. E., Kupfer, D. J., Eds.; Raven: New York, 1995; pp 505−517.

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